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Synthesis and Biological Activity of Peptide α-Ketoamide Derivatives as Proteasome Inhibitors
Pacifico, Salvatore; Ferretti, Valeria; Albanese, Valentina; Fantinati, Anna; Gallerani, Eleonora; Nicoli, Francesco; Gavioli, Riccardo; Zamberlan, Francesco; Preti, Delia; Marastoni, Mauro     dettagli >>
ACS MEDICINAL CHEMISTRY LETTERS
Vol. 10, No. 7, pp: 1086-1092, Anno: 2019

Naphthoquinone amino acid derivatives, synthesis and biological activity as proteasome inhibitors
Marastoni, Mauro; Trapella, Claudio; Scotti, Alessandra; Fantinati, Anna; Ferretti, Valeria; Marzola, Erika; Gallerani, Eleonora; Gavioli, Riccardo; Preti, Delia     dettagli >>
JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY
Vol. 32, No. 1, pp: 865-877, Anno: 2017

Studies of C-terminal naphthoquinone dipeptides as 20S proteasome inhibitors
Scotti, A; Trapella, Claudio; Ferretti, Valeria; Gallerani, Eleonora; Gavioli, Riccardo; Marastoni, Mauro     dettagli >>
JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY
Vol. 31, No. 3, pp: 456-463, Anno: 2016

Simultaneous inhibition of deubiquitinating enzymes (DUBs) and autophagy synergistically kills breast cancer cells
Vogel, Rachel Isaksson; Coughlin, Kathleen; Scotti, Alessandra; Iizuka, Yoshie; Anchoori, Ravi; Roden, Richard B. S.; Marastoni, Mauro; Bazzaro, Martina     dettagli >>
ONCOTARGET
Vol. 6, No. 6, pp: 4159-4170, Anno: 2015

Synthesis and activity of isoxazoline vinyl ester pseudopeptides as proteasome inhibitors.
Marastoni, Mauro; Scotti, Alessandra; Trapella, Claudio; Ferretti, Valeria; Sforza, Fabio; Gavioli, Riccardo     dettagli >>
JOURNAL OF PEPTIDE SCIENCE
Vol. 20, No. 4, pp: 258-265, Anno: 2014

C-terminal trans,trans-muconic acid ethyl ester partial retro-inverso pseudopeptides as proteasome inhibitors
Franceschini, C; Trapella, Claudio; Calia, R; Scotti, A; Sforza, F; Gavioli, Riccardo; Marastoni, Mauro     dettagli >>
JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY
Vol. 28, No. 1, pp: 1034-1039, Anno: 2013

Synthesis and biological properties of C-terminal vinyl ketone pseudotripeptides
Franceschini, C; Trapella, Claudio; Sforza, F; Gavioli, Riccardo; Marastoni, Mauro     dettagli >>
JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY
Vol. 28, No. 1, pp: 560-564, Anno: 2013

Proteasome inhibitors induce the presentation of an Epstein-Barr virus nuclear antigen 1-derived cytotoxic T lymphocyte epitope in Burkitt's lymphoma cells
Destro, Federica; Sforza, Fabio; Sicurella, Mariaconcetta; Marescotti, Diego; Gallerani, Eleonora; Baldisserotto, Anna; Marastoni, Mauro; Gavioli, Riccardo     dettagli >>
IMMUNOLOGY
Vol. 133, No. 1, pp: 105-114, Anno: 2011

Trypanocidal activity of peptidyl vinyl ester derivatives selective for inhibition of mammalian proteasome trypsin-like activity
Steverding, D.; Baldisserotto, Anna; Wang, X.; Marastoni, Mauro     dettagli >>
EXPERIMENTAL PARASITOLOGY
Vol. 128, No. 4, pp: 444-447, Anno: 2011

Synthesis and proteasome inhibition of N-allyl vinyl ester-based peptides
Baldisserotto, Anna; Franceschini, Christian; Scalambra, Franco; Trapella, Claudio; Marastoni, Mauro; Sforza, Fabio; Gavioli, Riccardo; Tomatis, Roberto     dettagli >>
JOURNAL OF PEPTIDE SCIENCE
Vol. 16, No. 11, pp: 659-663, Anno: 2010

Characterization of an human leucocyte antigen A2-restricted Epstein-Barr virus nuclear antigen-1-derived cytotoxic T-lymphocyte epitope
Marescotti, Diego; Destro, Federica; Baldisserotto, Anna; Marastoni, Mauro; Coppotelli, G.; Masucci, M.; Gavioli, Riccardo     dettagli >>
IMMUNOLOGY
Vol. 129, No. 3, pp: 386-395, Anno: 2010

α,β-Unsaturated N-Acylpyrrole Peptidyl Derivatives: New Proteasome Inhibitors
Baldisserotto, Anna; Ferretti, Valeria; Destro, Federica; Franceschini, Christian; Marastoni, Mauro; Gavioli, Riccardo; Tomatis, Roberto     dettagli >>
JOURNAL OF MEDICINAL CHEMISTRY
Vol. 53, No. 17, pp: 6511-6515, Anno: 2010

N-Terminal-prolonged vinyl ester-based peptides as selective proteasome b1 subunit inhibitors
Baldisserotto, Anna; Destro, Federica; Vertuani, Gianni; Marastoni, Mauro; Gavioli, Riccardo; Tomatis, Roberto     dettagli >>
BIOORGANIC & MEDICINAL CHEMISTRY
Vol. 17, No. 15, pp: 5535-5540, Anno: 2009

New cyclic peptide proteasome inhibitors
Baldisserotto, Anna; Marastoni, Mauro; Gavioli, Riccardo; Tomatis, Roberto     dettagli >>
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS
Vol. 19, No. 7, pp: 1966-1969, Anno: 2009

C-terminal constrained phenylalanine as a pharmacophoric unit in peptide-based proteasome inhibitors
Baldisserotto, Anna; Marastoni, Mauro; Lazzari, Ilaria; Trapella, Claudio; Gavioli, Riccardo; Tomatis, Roberto     dettagli >>
Editions Scientifique & Medical Elsevier:23 Rue Linois, F 75724 Paris Cedex 15 France:011 33 1 71724646, INTERNET: http://www.elsevier.fr, Fax: 011 33 1 71724664, EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY
Vol. 43, No. 7, pp: 1403-1411, Anno: 2008

Vinyl ester-based cyclic peptide proteasome inhibitors
Baldisserotto, Anna; Marastoni, Mauro; Fiorini, Stella; Pretto, Loretta; Ferretti, Valeria; Gavioli, Riccardo; Tomatis, Roberto     dettagli >>
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS
Vol. 18, No. 6, pp: 1849-1854, Anno: 2008

Peptide-based molecules for the production of positive charged liposomes and micelles
Cortesi, Rita; Marastoni, Mauro; Tomatis, Roberto; Menegatti, Enea; Esposito, Elisabetta; Nastruzzi, Claudio     dettagli >>
JOURNAL OF MICROENCAPSULATION
Vol. 25, No. 2, pp: 71-81, Anno: 2008

Glutamine vinyl ester proteasome inhibitors selective for trypsin-like (beta2) subunit
Baldisserotto, Anna; Marastoni, Mauro; Trapella, Claudio; Gavioli, Riccardo; Ferretti, Valeria; Pretto, Loretta; Tomatis, Roberto     dettagli >>
Editions Scientifique & Medical Elsevier:23 Rue Linois, F 75724 Paris Cedex 15 France:011 33 1 71724646, INTERNET: http://www.elsevier.fr, Fax: 011 33 1 71724664, EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY
Vol. 42, No. 5, pp: 586-592, Anno: 2007

Identification of CD8+ T cell epitopes within lytic antigens of human herpes virus 8
Ribechini, Eliana Melina; Fortini, Cinzia; Marastoni, Mauro; Traniello, S.; Spisani, Susanna; Monini, P.; Gavioli, Riccardo     dettagli >>
JOURNAL OF IMMUNOLOGY
Vol. 176, No. 1, pp: 923-930, Anno: 2006

Synthesis and biological evaluation of new vinyl ester pseudotripeptide proteasome inhibitors
Marastoni, Mauro; Baldisserotto, Anna; Trapella, Claudio; Gavioli, Riccardo; Tomatis, Roberto     dettagli >>
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY
Vol. 41, No. 8, pp: 978-984, Anno: 2006

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